Binding characteristics of a radiolabeled agonist and antagonist at central nervous system alpha noradrenergic receptors

Mol Pharmacol. 1977 May;13(3):454-73.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adrenergic alpha-Agonists / metabolism*
  • Adrenergic alpha-Antagonists / metabolism*
  • Animals
  • Binding Sites / drug effects
  • Binding, Competitive
  • Brain / metabolism*
  • Clonidine / metabolism*
  • Dioxanes / metabolism*
  • Dioxins / metabolism*
  • Ergot Alkaloids / pharmacology
  • Hydroxydopamines / pharmacology
  • In Vitro Techniques
  • Kinetics
  • Male
  • Norepinephrine / metabolism*
  • Phenethylamines / pharmacology
  • Phenyl Ethers / metabolism
  • Rats
  • Receptors, Adrenergic / metabolism*
  • Receptors, Adrenergic, alpha / drug effects
  • Receptors, Adrenergic, alpha / metabolism*
  • Time Factors

Substances

  • Adrenergic alpha-Agonists
  • Adrenergic alpha-Antagonists
  • Dioxanes
  • Dioxins
  • Ergot Alkaloids
  • Hydroxydopamines
  • Phenethylamines
  • Phenyl Ethers
  • Receptors, Adrenergic
  • Receptors, Adrenergic, alpha
  • Clonidine
  • Norepinephrine